#023 Dominic D'Agostino, Ph.D. on Modified Atkins Diet, Ketosis, Supplemental Ketones and More

Mar 23, 2016 Episode Page ↗
Overview

Dr. Dominic D'Agostino, an assistant professor at the University of South Florida, discusses nutritional ketosis, ketone supplementation, and their therapeutic and performance-enhancing effects. He highlights their potential for neurological disorders, cancer, and metabolic health, emphasizing the physiological adaptations and signaling roles of ketones.

At a Glance
28 Insights
1h 54m Duration
14 Topics
6 Concepts

Deep Dive Analysis

Introduction to Dr. D'Agostino's Metabolic Research

Defining and Measuring Nutritional Ketosis

Dietary Strategies for Achieving Ketosis: Classical vs. Modified Atkins

Impact of High-Fat Diets on Gut Health

Physiological Adaptations to Keto-Adaptation

Ketones as a Superior Fuel and Reactive Oxygen Species Reduction

Brain Energy Metabolism and Ketone Utilization

Ketones, Blood Flow, and Alzheimer's Disease

Therapeutic Potential of Ketone Supplementation

Ketones and Cancer Treatment in Animal Models

Metformin's Role in Cancer Prevention and Longevity

Gluconeogenesis and Glucose Production in Ketosis

Glutamine's Dual Role in Cancer and Gut Health

Future of Ketone Supplements and Ketogenic Food Products

Nutritional Ketosis

Nutritional ketosis is defined as achieving and sustaining blood ketone levels above 0.5 millimolar, ideally between 1 and 3 millimolar. This state is driven by the suppression of the hormone insulin, which in turn drives hepatic ketogenesis.

Classical Ketogenic Diet

This is a very strict diet, typically comprising 85-90% fat, 8-10% protein, and minimal carbohydrates. It was originally heavily based on dairy fat and used for drug-resistant epilepsy, but is challenging to follow due to its restrictive nature.

Modified Atkins Diet

A more liberal approach to the ketogenic diet, consisting of roughly 65-70% fat, 20-30% protein, and 5-10% carbohydrates. It has shown similar therapeutic potency to the classical ketogenic diet for drug-resistant epilepsy, making it more accessible.

Keto-adaptation

This is a physiological process where the body adapts to primarily using fatty acids and ketones for fuel instead of glucose. Over time, it leads to an upregulation of ketone transport and utilization mechanisms, as well as an increased oxidative capacity of cells.

Glucose Sparing

When the brain utilizes ketones as a primary energy source, it can 'spare' glucose, allowing it to be shunted into other metabolic pathways. This includes the pentose phosphate pathway, which is crucial for generating NADPH, important for glutathione recycling and dealing with stress.

Metabolic Theory of Cancer

This theory proposes that cancer originates from progressive damage to mitochondrial oxidative phosphorylation, leading to impaired energy status in the cell. This energetic crisis then triggers the nucleus to activate oncogenes, transforming a normal cell into a cancer cell with a Warburg (glycolytic) phenotype.

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What is nutritional ketosis and how is it defined?

Nutritional ketosis is defined as achieving and sustaining blood ketone levels above 0.5 millimolar, ideally between 1 and 3 millimolar, which can be measured using blood ketone devices.

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What are the typical macronutrient ratios for a classical ketogenic diet?

A classical ketogenic diet is typically very high in fat (85-90%), moderate to low in protein (8-10%), and very low in carbohydrates, often based on dairy fat.

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How does the Modified Atkins Diet differ from the classical ketogenic diet?

The Modified Atkins Diet is more liberal, consisting of roughly 65-70% fat, 20-30% protein, and 5-10% carbohydrates, making it more accessible while retaining therapeutic potency.

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Can a high-fat diet harm the gut microbiome?

While high-fat diets in animal studies can induce endotoxin release, a 'well-formulated' ketogenic diet with diverse raw vegetables can actually improve gut health and microbiome diversity by feeding different bacteria.

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How do ketones reduce reactive oxygen species (ROS) production?

Ketones, particularly beta-hydroxybutyrate, lead to oxidized ubiquinone (Q), making it less available to react with molecular oxygen in the electron transport chain, thus producing less superoxide anion.

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Why might the brain prefer ketones as a fuel source in certain conditions?

In contexts like aging, traumatic brain injury, pathology, or stress (e.g., hypoglycemia), the brain may prefer ketones due to impaired brain glucose metabolism, such as issues with GLUT3 transporters or pyruvate dehydrogenase complex.

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Do ketone supplements offer similar benefits to a ketogenic diet or fasting?

Yes, studies in animal models have shown that ketone supplementation can prevent CNS oxygen toxicity and significantly increase survival time in metastatic cancer models, even on a high-carbohydrate diet.

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How does metformin relate to cancer prevention?

Metformin, a diabetes drug, has been shown in retrospective studies to reduce the risk of certain cancers (e.g., pancreatic cancer by 62% in type 2 diabetics) and is being studied as a potential preventative therapy due to its effects on AMP kinase, mTOR, and insulin signaling.

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Is it safe to take glutamine supplements if you have cancer?

For GI cancers and liver cancer, it is advisable to avoid or minimize glutamine supplementation and high glutamine-containing foods, as these cells may utilize glutamine for growth. For other cancers, if systemic treatments impair gut function, a small amount of glutamine might be helpful for gut repair.

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Do ketones help preserve muscle mass during a ketogenic diet?

Yes, ketones are considered anti-catabolic and protein-sparing, meaning they help protect gluconeogenic amino acids and skeletal muscle from being degraded, especially when ample fat is consumed to provide sufficient fuel.

1. Measure Blood Ketones

To confirm you are in a state of ketosis, measure your blood ketones and aim for levels between 1 and 3 millimolar, with a minimum of 0.5 millimolar. This helps verify if a ketogenic diet or intervention is effective.

2. Prioritize Diverse Raw Vegetables

To optimize gut health and microbiome diversity on a ketogenic diet, ensure you include a diverse variety of raw vegetables as carbohydrate sources.

3. Optimize Carb & Fat Sources

Beyond macronutrient ratios, optimize your ketogenic diet by focusing on the sources of fats, the type of protein, and the quality and type of carbohydrates, as these factors are crucial for individual health and gut microbiome diversity.

4. Avoid High Protein on Keto

When following a ketogenic diet, ensure your protein intake is moderate to low, not high, as many people mistakenly consume a high-protein, moderate-fat diet instead of a true ketogenic diet. High protein can hinder ketosis.

5. Consult a Savvy Dietitian

If you plan to try a ketogenic diet, start by consulting a savvy dietitian who can tailor and tweak the diet to your specific needs, as their experience is invaluable.

6. Consider Modified Atkins Diet

For a more accessible approach to therapeutic ketosis, consider the Modified Atkins Diet, which is 65-70% fat, 20-30% protein, and 5-10% carbohydrates, allowing for more protein and incorporating medium-chain fatty acids while maintaining therapeutic potency.

7. Personalize Ketogenic Diet

Tailor your ketogenic diet to your individual sensitivities, such as avoiding dairy or nuts if you have allergies or intolerances, to optimize your personal health and adherence.

8. Include Liberal Vegetables on Keto

To support gut health while on a ketogenic diet, ensure your diet includes a liberal amount of vegetables, as this has been associated with better gut health for some individuals.

9. Use Vegetables to Slow Digestion

Incorporate vegetables into your ketogenic diet as carriers for fat, as they help slow protein digestion, minimize insulin spikes, and aid in maintaining ketosis.

10. Use MCT Powder for Mild Ketosis

To achieve a mild state of ketosis with better GI tolerance than liquid MCT oil, use MCT powder, consuming 4-8 scoops daily mixed with water, coffee, or tea.

11. Prioritize Whole Foods with Ketones

Even when using ketone supplements, prioritize a whole-food diet free of refined crap and processed foods, as a poor diet will significantly diminish the benefits of ketones.

12. Cycle Metabolic Strategies for Flexibility

To promote metabolic flexibility and enhance the long-term effectiveness of interventions, cycle between different dietary strategies like a paleo diet, a low-carb ketogenic diet, and intermittent fasting on occasional days, rather than strictly adhering to one continuously.

13. Maintain Ketosis to Preserve Muscle

Maintain a state of ketosis to leverage its anti-catabolic and protein-sparing effects, which help protect gluconeogenic amino acids and skeletal muscle from degradation.

14. Ensure Ample Fat on Ketogenic Diet

When on a ketogenic diet, ensure you consume ample amounts of fat, as insufficient fat intake can lead to a more catabolic state.

15. Use Ketones for Appetite Control

Utilize ketones to help control appetite, as they have a satiating effect by sending energy to the brain and can shut off hypoglycemic triggers that lead to food cravings or binges.

16. Consider Ketogenic Intermittent Fasting

For potential cancer prevention or post-treatment care, consider a ketogenic intermittent fasting protocol where you consume ketogenic fats and ketone supplements for 20 hours, followed by a four-hour window to eat a well-balanced ketogenic meal rich in vegetables and healthy fats and protein.

17. Metformin for Cancer Prevention (Consult Doctor)

Discuss with your doctor the potential of metformin as a preventative therapy, especially if you are at risk for certain cancers like pancreatic cancer, given studies showing a significant reduction in risk for type 2 diabetics taking the drug.

18. Monitor B12 with Metformin

If taking metformin, be aware of potential vitamin B12 deficiency and consider supplementing with a sublingual form or B12 injections, especially as B12 absorption decreases with age.

19. Enhance Drug Delivery with Ketosis

If taking drugs that need to cross the blood-brain barrier (e.g., chemotherapeutics), consider inducing ketosis through fasting or a ketogenic diet, as this may increase blood-brain barrier permeability and facilitate faster drug transport.

20. Avoid Glutamine for GI/Liver Cancer

If you have gastrointestinal or liver cancer, avoid supplementing with glutamine and minimize high glutamine-containing foods, as these cancers may utilize glutamine for growth.

21. Glutamine for Impaired GI Function (Non-GI Cancer)

If you have impaired GI function due to systemic treatments (e.g., for a brain tumor) and do not have GI or liver cancer, a small amount (5-10 grams) of oral glutamine may be helpful to repair your gut.

22. Lower Glutamine on Ketogenic Diet

A classical ketogenic diet (low to moderate protein) can help lower blood glutamine levels, which may be beneficial in certain cancer contexts.

23. Select Low-Glutamine Protein Sources

To further suppress glutamine levels, select protein food sources that are lower in glutamine and consider avoiding glutamine supplementation, opting instead for supplements high in essential amino acids (excluding glutamine).

24. Lauric Acid Suppresses Hunger

Consider consuming lauric acid (C12) as it has been shown to suppress ghrelin, a hunger hormone, in the gut.

25. Classical Ketogenic Diet Ratios

To achieve nutritional ketosis, a classical ketogenic diet typically involves a 4:1 or 3:1 ratio of fat to combined carbohydrates and protein, often translating to 85-90% fat, 8-10% protein, and minimal carbohydrates, historically relying heavily on dairy fat.

26. Ketone Supplements for Cancer (Research)

Research suggests that ketone supplementation, even on a high-carbohydrate diet, can reduce tumor growth and proliferation and increase survival time in aggressive metastatic cancer models, indicating potential anti-cancer effects.

27. Avoid Antioxidant Supplements for Cancer (Research)

Studies suggest that giving mice supplemental vitamin E or N-acetylcysteine (NAC), which potently sequester reactive oxygen species, can actually allow tumors to grow faster, implying caution with antioxidants in cancer contexts.

28. Ketone Esters for Potent Ketosis (Future)

For a powerful form of exogenous ketones, look for ketone esters (currently in development for human use) which have shown significant effects, such as preventing CNS oxygen toxicity.

Pretty much every neurological disorder is some way linked to a metabolic dysregulation.

Dr. Dominic D'Agostino

Ketones are more than just the metabolite. They're more than just an energy metabolite the brain can use, but they are... metabolites, especially beta-hydroxybutyrate, are very powerful signaling molecules.

Dr. Dominic D'Agostino

The ketogenic diet is not a high-protein diet. It's actually moderate to low-protein diet, and most people don't understand that.

Dr. Dominic D'Agostino

If Q is oxidized, then you have less availability for that electron to react with molecular oxygen in the metabolic pathway. So, you would produce less superoxide anion, which is your precursor to more reactive oxygen species.

Dr. Dominic D'Agostino

The stability of the nuclear genome is tightly regulated to the energetic state of the cell.

Dr. Dominic D'Agostino

Ketones, we know undoubtedly they have anti-cancer effects, and it could be maybe through their expression of their gene expression as a histone deacetylase inhibitor.

Dr. Dominic D'Agostino

Metabolic interventions tend to work best when you cycle them, I think.

Dr. Dominic D'Agostino

If you're in a state of ketosis, you're protecting gluconeogenic amino acids and skeletal muscle from being degraded.

Dr. Dominic D'Agostino

Modified Atkins Diet for Therapeutic Ketosis

Dr. Dominic D'Agostino (referencing Eric Kosoff's work)
  1. Consume roughly 65-70% of total calories from fat.
  2. Consume about 20-30% of total calories from protein.
  3. Limit carbohydrates to no more than 5-10% of total calories.
  4. Incorporate medium-chain fatty acids into the diet.
  5. Optimize the diversity of carbohydrate sources, primarily from raw vegetables, to support gut health.

Ketogenic Intermittent Fasting (Proposed)

Dr. Dominic D'Agostino
  1. Consume ketogenic fats and ketone supplements throughout a 20-hour fasting window.
  2. Eat a well-balanced ketogenic meal, rich in vegetables, high in fats, and protein, within a 4-hour eating window.
0.5 millimolar
Minimum blood ketone level for nutritional ketosis At the very least; ideally between 1 and 3 millimolar
85% to 90%
Fat content in classical ketogenic diet Of total calories
8% to 10%
Protein content in classical ketogenic diet Of total calories, very minimal carbohydrates
65% to 70%
Fat content in Modified Atkins Diet Of total calories
20% to 30%
Protein content in Modified Atkins Diet Of total calories
5% to 10%
Carbohydrate content in Modified Atkins Diet Of total calories, no more than
Over 500%
Delay in CNS oxygen toxicity with ketone ester Observed in a rat model using an oral ketone ester supplement
50% to 60%
Increase in survival time with ketone supplementation in metastatic cancer model Observed in animals on a high-carbohydrate diet supplemented with ketone ester
30% to 40%
Increase in brain blood flow with ketone bodies Previous work has shown this effect
62%
Reduction in pancreatic cancer risk for type 2 diabetics taking metformin Based on studies of people taking metformin
7% to 10%
Percentage of cancers linked to hereditary effect Estimate of cancers originating from hereditary factors
2 millimolar
Typical glutamine level used in in vitro studies For glutamine withdrawal experiments
Up to 40% or 50%
Percentage of people with GI tolerability issues for liquid MCTs When taking a big dose to achieve sustainable ketosis